Patent · US Active

Small molecule inhibitors of PARP activity

US8513433B2 · kind B2 · utility

45Cited by
1References
21Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 2, 2010
Grant dateAug 20, 2013
Priority date
Expiry dateJul 2, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D401/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds and pharmaceutical compositions are provided that inhibit the activity of poly ADP-ribose synthetase (PARP). Such compounds are useful in the treatment of various diseases, conditions and injuries such as stroke, myocardial infarction, ischemia-perfusion injury in various organs, traumatic brain injury, atherosclerosis, inflammatory diseases and cancer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.