Patent · US Active

Cyclosporin derivatives for treating inflammatory diseases and conditions

US8524671B2 · kind B2 · utility

2Cited by
8References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 21, 2010
Grant dateSep 3, 2013
Priority date
Expiry dateJun 6, 2031

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/08
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides a method for the treatment of inflammatory diseases and/or conditions, e.g. allergic conjunctivitis, uveitis or phacoanaphylactic endophthalmitis in an eye of a mammal, said method comprising administering to said mammal in need of treatment a therapeutically effective amount of a novel cyclosporin A derivative selected from the group consisting of compounds represented by the formula:wherein R1 is S-Alk-R wherein Alk is an alkylene linkage, preferably a methylene or poly methylene linkage, or a polyalkenylene linkage, e.g. a C3 to C6 alkenylenyl linkage and R is a hydrogen or a unsubstituted or substituted hydrocarbyl group.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.