Patent · US Active

Proteasome inhibitors and methods of using the same

US8546608B2 · kind B2 · utility

2Cited by
31References
3Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 30, 2011
Grant dateOct 1, 2013
Priority date
Expiry dateSep 30, 2031

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F5/025
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides boronic acid compounds, boronic esters, and compositions thereof that can modulate apoptosis such as by inhibition of proteasome activity. The compounds and compositions can be used in methods of inducing apoptosis and treating diseases such as cancer and other disorders associated directly of indirectly with proteasome activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.