Patent · US Active

Pyrazolopyrimidines and related heterocycles as CK2 inhibitors

US8575177B2 · kind B2 · utility

8Cited by
1References
40Claims
0Family size

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Inventors

Key dates

Filing dateNov 15, 2010
Grant dateNov 5, 2013
Priority date
Expiry dateJan 21, 2031

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides compounds that inhibit protein kinase CK2 activity (CK2 activity), and compositions containing such compounds. These compounds and compositions are useful for treating proliferative disorders such as cancer, as well as other kinase-associated conditions including inflammation, pain, and certain immunological disorders, and have the following general formula:

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.