Patent · US Active

Solid dispersion formulations and methods of use thereof

US8591944B2 · kind B2 · utility

1Cited by
63References
29Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 7, 2012
Grant dateNov 26, 2013
Priority date
Expiry dateMar 7, 2032

Classification

  • Technology area (CPC B)Performing Operations; Transporting
  • CPC primaryB29C48/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to formulations and methods for increasing the bioavailability of 1-(4-benzhydrylpiperazin-1-yl)-3,3-diphenylpropan-1-one, 1-(3,3-diphenylpropanoyl)piperazine, or a salt thereof. In particular, the formulation can include one or more pharmaceutically acceptable matrix polymers to form a solid dispersion, e.g., a spray dried dispersion or a hot melt extrusion.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.