Method for the regioselective synthesis of 1-alky1-3-haloalkyl-pyrazole-4-carboxylic acid derivatives
US8629288B2 · kind B2 · utility
5Cited by
4References
11Claims
0Family size
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Key dates
| Filing date | Feb 12, 2009 |
| Grant date | Jan 14, 2014 |
| Priority date | — |
| Expiry date | Feb 12, 2029 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D231/14
- WIPO fieldOrganic fine chemistry
- WIPO sectorChemistry
Abstract
The present invention relates to a process for the regioselective synthesis of 1-alkyl-3-halo-alkylpyrazole-4-carboxylic acid derivatives by cyclization of 2,3-disubstituted acrylic acid derivatives, and to the hydrazones formed as intermediates in the process.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.