Patent · US Active

Method for the regioselective synthesis of 1-alky1-3-haloalkyl-pyrazole-4-carboxylic acid derivatives

US8629288B2 · kind B2 · utility

5Cited by
4References
11Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 12, 2009
Grant dateJan 14, 2014
Priority date
Expiry dateFeb 12, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D231/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a process for the regioselective synthesis of 1-alkyl-3-halo-alkylpyrazole-4-carboxylic acid derivatives by cyclization of 2,3-disubstituted acrylic acid derivatives, and to the hydrazones formed as intermediates in the process.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.