Imidazolo-, oxazolo-, and thiazolopyrimidine modulators of TRPV1
US8637527B2 · kind B2 · utility
1Cited by
13References
19Claims
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Key dates
| Filing date | Sep 12, 2012 |
| Grant date | Jan 28, 2014 |
| Priority date | — |
| Expiry date | Sep 12, 2032 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D498/04
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Certain TRPV1-modulating imidazolo-, oxazolo-, and thiazolopyrimdine compounds are described. The compounds may be used in pharmaceutical compositions and methods for treating disease states, disorders, and conditions mediated by TRPV1 activity, such as pain, arthritis, itch, cough, asthma, or inflammatory bowel disease.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.