Vanilloid receptor ligands, pharmaceutical compositions containing them, process for making them, and use thereof for treating pain and other conditions

US8642775B2 · kind B2 · utility

Assignee

• Gruenenthal GmbH · DE

Inventors

• Robert Frank · Aachen, DE
• Gregor Bahrenberg · Monschau, DE
• Thomas Christoph · Aachen, DE
• Klaus Schiene · Goldkronach, DE
• Jean De Vry · Stolberg, DE
• Derek Saunders · Aachen, DE
• Michael Przewosny · Aachen, DE
• Bernd Sundermann · Aachen, DE
• Jewoo Lee · Seojong-myeon, KR

Key dates

• Filing date: Apr 15, 2008
• Grant date: Feb 4, 2014
• Expiry date: Sep 12, 2028

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D213/70
• WIPO field: Pharmaceuticals
• WIPO sector: Chemistry

Abstract

Vanilloid receptor ligand compounds corresponding to formula I:a process for producing such compounds, pharmaceutical compositions containing them, and the use of such compounds to treat pain and various other vanilloid receptor mediated conditions.