Patent · US Active

Wet granulation using a water sequestering agent

US8652492B2 · kind B2 · utility

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Key dates

Filing dateJan 10, 2013
Grant dateFeb 18, 2014
Priority date
Expiry dateJan 10, 2033

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P37/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed are tablets comprising hydrolytically stable formulations of (6-(5-fluoro-2-(3,4,5-trimethoxyphenylamino)pyrimidin-4-ylamino)-2,2-dimethyl-3-oxo-2H-pyrido[3,2-b][1,4]oxazin-4(3H)-yl)methyl phosphate disodium salt (Compound 1) prepared by a wet granulation process.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.