Patent · US Active

Crystalline ingenol mebutate

US8653133B2 · kind B2 · utility

2Cited by
0References
27Claims
0Family size

Assignee

Inventor

Key dates

Filing dateApr 18, 2011
Grant dateFeb 18, 2014
Priority date
Expiry dateOct 26, 2031

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02A50/30
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to a novel crystalline form of ingenol mebutate, methods of preparation thereof, and to its use. More specifically, the invention relates to the conversion of amorphous ingenol mebutate (ingenol-3-angelate, PEP005) to a crystalline form, which was characterized by single crystal X-Ray crystallography (XRC), attenuated total reflectance Fourier transform infrared (FTIR-ATR) spectroscopy and Differential Scanning calorimetry (DSC).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.