Patent · US Active

3,5-diamino-6-chloro-pyrazine-2-carboxylic acid derivatives and their use as epithelial sodium channel blockers for the treatment of airway diseases

US8664228B2 · kind B2 · utility

6Cited by
2References
3Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 11, 2009
Grant dateMar 4, 2014
Priority date
Expiry dateAug 3, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound of Formula Iin free or salt or solvate form, where R1, R2, R3, R4, R5, R6, R7, R8 and R9 have the meanings as indicated in the specification, is useful for treating diseases which respond to the blockade of the epithelial sodium channel. Pharmaceutical compositions that contain the compounds and processes for preparing the compounds are also described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.