Patent · US Active

Process for the preparation of (poly) aminoalkylaminoacetamide derivatives of epipodophyllotoxin useful for their applications in therapeutics as anticancer agent

US8664409B2 · kind B2 · utility

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1References
18Claims
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Key dates

Filing dateSep 23, 2008
Grant dateMar 4, 2014
Priority date
Expiry dateJul 28, 2029

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a new process for the preparation of (poly)aminoalkylaminoacetamide derivatives of epipodophyllotoxin and salts thereof, characterized in that it comprises a step of peptide coupling of 4-amino-4′-demethylepipodophyllotoxin with an amine-containing reactant having protecting groups.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.