Patent · US Active

Cannabinoid receptor antagonists/inverse agonists useful for treating disease conditions, including metabolic disorders and cancers

US8680131B2 · kind B2 · utility

2Cited by
9References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 24, 2013
Grant dateMar 25, 2014
Priority date
Expiry dateJul 24, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D231/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides novel, diastereomeric pyrazolines that are useful as cannabinoid receptor blockers and pharmaceutical compositions thereof and methods of using the same for treating obesity, diabetes, inflammatory disorders, cardiometabolic disorders, hepatic disorders, and/or cancers.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.