Patent · US Active

D2 antagonists, methods of synthesis and methods of use

US8691836B2 · kind B2 · utility

2Cited by
4References
14Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 17, 2011
Grant dateApr 8, 2014
Priority date
Expiry dateApr 24, 2032

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02A50/30
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Provided are D2 or D3 antagonist compounds and pharmaceutical compositions of formula Iand pharmaceutically acceptable salts thereof, or isomers thereof, wherein R1, R2 and R3 are as defined herein. The invention further comprises methods for making the compounds of the invention and methods for the treatment of conditions mediated by the dopamine D2 or D3 receptor from the compounds of the invention.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.