Thiophenyl and pyrrolyl azepines as serotonin 5-HT2C receptor ligands and uses thereof
US8716276B2 · kind B2 · utility
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3Claims
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Key dates
| Filing date | Jan 12, 2011 |
| Grant date | May 6, 2014 |
| Priority date | — |
| Expiry date | Mar 4, 2032 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D495/06
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The present invention generally relates to a series of compounds, to pharmaceutical compositions containing the compounds, and to use of the compounds and compositions as therapeutic agents. More specifically, compounds of the present invention are thiophenyl and pyrrolyl azepine compounds. These compounds are serotonin receptor (5-HT2c) ligands and are useful for treating diseases, disorders, and conditions wherein modulation of the activity of serotonin receptors (5-HT2c) is desired (e.g. addiction, anxiety, depression, obesity, and others).
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.