Patent · US Active

Pharmaceutical compositions containing quinazoline derivatives for treating as serotonin receptor antagonist

US8748422B2 · kind B2 · utility

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10Claims
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Assignee

Inventors

Key dates

Filing dateAug 21, 2008
Grant dateJun 10, 2014
Priority date
Expiry dateJan 16, 2031

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P25/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to a pharmaceutical composition containing one or more quinazoline compounds as an active ingredient, which has antagonistic activity against serotonin 5-HT3A and is effective for the prevention and treatment of central nervous system (CNS) diseases, including emesis, nausea, alcoholism, drug abuse, depression, compulsive neurosis, anxiety, seizure, Alzheimer's disease, Parkinson's disease, Huntington's chorea, psychosis, schizophrenia, suicidal tendency, sleep disorder, appetite disorder and migraine.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.