Patent · US Active

N-containing heterocyclic compounds

US8765755B2 · kind B2 · utility

3Cited by
2References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 5, 2012
Grant dateJul 1, 2014
Priority date
Expiry dateDec 5, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to N-containing heterocyclic compounds that are inhibitors of protein kinases including JAK kinases. In particular, the compounds are selective for JAK1, JAK2, JAK3 or TYK2 kinases and combinations thereof such as JAK1 and JAK2. The kinase inhibitors can be used in the treatment of kinase associated diseases such as immunological and inflammatory diseases including organ transplants; hyperproliferative diseases including cancer and myeloproliferative diseases; viral diseases; metabolic diseases; and vascular diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.