Carbamoyl derivatives of bicyclic carbonylamino-pyrazoles as prodrugs
US8809337B2 · kind B2 · utility
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3Claims
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Key dates
| Filing date | Sep 28, 2012 |
| Grant date | Aug 19, 2014 |
| Priority date | — |
| Expiry date | Sep 28, 2032 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D497/04
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
There are provided bicyclic carbonylamino-pyrazoles of formula (I), wherein the variables are as specified in the claims, for use as medicament, in particular for the treatment of diseases due to the malfunctioning of protein kinases (PKs), such as cancer, pharmaceutical compositions comprising such carbamoyl derivatives, and their use as prodrugs of therapeutically active agents. Method of treatment and some new bicyclic carbonylamino-pyrazoles are also object of the present invention.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.