Patent · US Active

Agents for treating disorders involving modulation of ryanodine receptors

US8853198B2 · kind B2 · utility

4Cited by
4References
29Claims
0Family size

Assignees

Inventors

Key dates

Filing dateNov 11, 2013
Grant dateOct 7, 2014
Priority date
Expiry dateNov 11, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D285/36
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to 1,4-benzothiazepine derivatives and their use to treat conditions, disorders and diseases associated with ryanodine receptors (RyRs) that regulate calcium channel functioning in cells. The invention also discloses pharmaceutical compositions comprising the compounds and uses thereof to treat diseases and conditions associated with RyRs, in particular cardiac, musculoskeletal and central nervous system (CNS) disorders.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.