Patent · US Active

Inhibitor of analgesic tolerance

US8865731B2 · kind B2 · utility

11Cited by
8References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 29, 2009
Grant dateOct 21, 2014
Priority date
Expiry dateSep 14, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Provided are: an agent for suppressing an undesirable effect of an opioid-type analgesic (opioid), which comprises a compound having adenosine A2A receptor antagonistic activity or a pharmaceutically acceptable salt thereof as an active ingredient; the agent for suppressing an undesirable effect of an opioid-type analgesic (opioid), wherein the undesirable effect of the opioid-type analgesic (opioid) is analgesic tolerance or constipation; the agent for suppressing an undesirable effect of an opioid-type analgesic (opioid), wherein the undesirable effect of the opioid-type analgesic (opioid) is analgesic tolerance; and the like.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.