Patent · US Active

Crystalline pharmaceutical and methods of preparation and use thereof

US8871935B2 · kind B2 · utility

2Cited by
63References
3Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 11, 2012
Grant dateOct 28, 2014
Priority date
Expiry dateJan 7, 2033

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K47/183
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Novel crystalline polymorphic forms, Forms A, B, C, D, and E of a compound of Formula I, which has been found to be a potent inhibitor of LFA-1, are disclosed. Methods of preparation and uses thereof in the treatment of LFA-1 mediated diseases are also disclosed in this invention.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.