Patent · US Active

Polymorphs of Dasatinib, preparation methods and pharmaceutical compositions thereof

US8884013B2 · kind B2 · utility

16Cited by
1References
10Claims
0Family size

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Key dates

Filing dateJan 31, 2011
Grant dateNov 11, 2014
Priority date
Expiry dateJan 31, 2031

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Polymorph I of dasatinib monohydrate and Polymorph II of dasatinib, their preparation methods and pharmaceutical compositions containing the same are provided. These polymorphs have better physicochemical properties, are more stable and are more suitable for industrial scale production.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.