6-amino quinazoline or 3-cyano quinoline derivatives, preparation methods and pharmaceutical uses thereof
US8901140B2 · kind B2 · utility
Assignees
Inventors
Key dates
| Filing date | Aug 26, 2010 |
| Grant date | Dec 2, 2014 |
| Priority date | — |
| Expiry date | Dec 10, 2030 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07F9/65128
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
6-amino quinazoline or 3-cyano quinoline derivatives, preparation methods and pharmaceutical uses thereof are disclosed. Specifically, the present disclosure discloses novel 6-amino quinazoline or 3-cyano quinoline derivatives presented by general formula (I), or tautomers, enantiomers, diastereomers, racemates or pharmaceutically acceptable salts thereof, or metabolites, metabolic precursors or prodrugs thereof, and their uses as treatment agents especially as protein kinase inhibitors, in which each substitutent group of general formula (I) is as defined in the specification.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.