Patent · US Active

6-amino quinazoline or 3-cyano quinoline derivatives, preparation methods and pharmaceutical uses thereof

US8901140B2 · kind B2 · utility

3Cited by
0References
17Claims
0Family size

Assignees

Inventors

Key dates

Filing dateAug 26, 2010
Grant dateDec 2, 2014
Priority date
Expiry dateDec 10, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/65128
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

6-amino quinazoline or 3-cyano quinoline derivatives, preparation methods and pharmaceutical uses thereof are disclosed. Specifically, the present disclosure discloses novel 6-amino quinazoline or 3-cyano quinoline derivatives presented by general formula (I), or tautomers, enantiomers, diastereomers, racemates or pharmaceutically acceptable salts thereof, or metabolites, metabolic precursors or prodrugs thereof, and their uses as treatment agents especially as protein kinase inhibitors, in which each substitutent group of general formula (I) is as defined in the specification.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.