Patent · US Active

Tricyclic derivatives, process for their preparation and their use as kinase inhibitors

US8916577B2 · kind B2 · utility

2Cited by
0References
21Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 19, 2012
Grant dateDec 23, 2014
Priority date
Expiry dateJan 19, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D498/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

New substituted tricyclic compounds of formula (I) are described, wherein R1, R2, X, Y, Z are herein defined, having protein kinase inhibiting activity. The invention includes methods to prepare the compounds of formula (I), pharmaceutical compositions containing them, and their use in therapy, in particular for the treatment of diseases caused by and/or associated with dysregulated activity of protein kinase.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.