Patent · US Active

Thio derivatives bearing lactams as potent HDAC inhibitors and their uses as medicaments

US8927533B2 · kind B2 · utility

1Cited by
1References
11Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 17, 2012
Grant dateJan 6, 2015
Priority date
Expiry dateSep 17, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D401/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to novel amide compounds of Formula (I), and their use as anti-tumoral and pro-apoptotic agents. The invention includes the use of such compounds in medicine, in relation to cancer disease as well as other diseases where an inhibition of HDAC is responsive, and the pharmaceutical composition containing such compounds.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.