Patent · US Active

Unsaturated nitrogen heterocyclic compounds useful as PDE10 inhibitors

US8957073B2 · kind B2 · utility

10Cited by
2References
31Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 11, 2011
Grant dateFeb 17, 2015
Priority date
Expiry dateMar 21, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Unsaturated nitrogen heterocyclic compounds of formula (I):as defined in the specification, compositions containing them, and processes for preparing such compounds. Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, Huntington's Disease, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obsessive-compulsive disorder, and the like.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.