Patent · US Active

Antitumor agent for thyroid cancer

US9006256B2 · kind B2 · utility

42Cited by
70References
6Claims
0Family size

Assignee

Inventor

Key dates

Filing dateApr 8, 2011
Grant dateApr 14, 2015
Priority date
Expiry dateJun 18, 2031

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12Q2600/106
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides pharmaceutical compositions and therapeutic methods for treating diseases such as multiple endocrine neoplasia type IIA, multiple endocrine neoplasia type IIB, familial medullary thyroid carcinoma, thyroid carcinoma, papillary thyroid carcinoma, sporadic medullary thyroid carcinoma, Hirschsprung disease, pheochromocytoma, parathyroid hyperplasia and mucosal neuromas of the gastrointestinal tract. The therapeutic methods and pharmaceutical compositions use a RET kinase inhibiting substance, such as 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)-7-methoxy-6-quinolinecarboxamide and pharmacologically acceptable salts thereof, and involve a step of administering the RET kinase inhibiting substance to a patient.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.