Patent · US Active

Acetaminophen conjugates, compositions and methods of use thereof

US9024055B2 · kind B2 · utility

6Cited by

8References

9Claims

0Family size

Assignee

Acorda Therapeutics, Inc. · US

Inventors

Keith R. Bley · Menlo Park, US
Bernd Jandeleit · Menlo Park, US

Key dates

Filing date	Sep 21, 2012
Grant date	May 5, 2015
Priority date	—
Expiry date	Sep 21, 2032

Classification

Technology area (CPC C)Chemistry; Metallurgy
CPC primaryC07C313/04
WIPO fieldPharmaceuticals
WIPO sectorChemistry

Abstract

Acetaminophen conjugates are provided, which have an acetaminophen moiety covalently linked to a second moiety. The conjugates provided may have one or more advantageous properties, including increased water solubility as compared to acetaminophen, reduced toxicity profile as compared to acetaminophen and an altered pharmacokinetic profile. Formulations comprising the conjugates are also provided, as are methods of using the conjugates and kits comprising the conjugates.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.