Patent · US Active

Antioxidant nanosphere comprising [1,2]-dithiolane moieties

US9028874B2 · kind B2 · utility

1Cited by
32References
26Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 30, 2008
Grant dateMay 12, 2015
Priority date
Expiry dateApr 20, 2031

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K9/0014
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention is directed to multiple a-lipoic acid-containing hydrophobic compounds (mALAs) capable of acting as scavengers of free radicals, metals and reactive oxygen species (ROS). Methods of synthesizing novel antioxidant mALAs, spontaneous emulsification or nanoprecipitaion thereof to produce antioxidant nanospheres and their use in preventing or treating diseases or conditions caused by oxidative stress and other free radical mediated conditions are also described. Another aspect of this invention is the use of these antioxidant nanospheres for the preparation of antioxidant particulate delivery system of therapeutic agents.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.