Patent · US Active

Heterocyclyl pyrazolopyrimidine analogues as selective JAK inhibitors

US9040545B2 · kind B2 · utility

0Cited by
0References
5Claims
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Assignee

Inventors

Key dates

Filing dateAug 12, 2011
Grant dateMay 26, 2015
Priority date
Expiry dateNov 12, 2031

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D519/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to compounds of formula (I)wherein X1 to X5, Y, Z1 to Z3, and R have the meaning as cited in the description and the claims. Said compounds are useful as JAK inhibitors for the treatment or prophylaxis of immunological, inflammatory, autoimmune, allergic disorders, and immunologically-mediated diseases. The invention also relates to pharmaceutical compositions including said compounds, the preparation of such compounds as well as the use as medicaments.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.