Patent · US Active

Glycosylated aminocoumarins and methods of preparing and uses of same

US9045517B2 · kind B2 · utility

0Cited by
2References
5Claims
0Family size

Assignee

Inventor

Key dates

Filing dateOct 17, 2011
Grant dateJun 2, 2015
Priority date
Expiry dateFeb 17, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12P19/605
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

There is provided a method of glycosylating an aminocoumarin compound comprising conjugating a sugar to the 4′-OH position of the core of the aminocoumarin compound. Also provided is an aminocoumarin compound glycosylated at the 4′-OH position of the core of the aminocoumarin compound. Further aspects of this invention provide this compound for use in therapy, more particularly for use as an antibiotic, or in anticancer treatment.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.