Patent · US Active

Pyrazine derivatives as ENaC blockers

US9050339B2 · kind B2 · utility

2Cited by
3References
8Claims
0Family size

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Key dates

Filing dateOct 22, 2012
Grant dateJun 9, 2015
Priority date
Expiry dateJul 31, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/10
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of Formula I:and pharmaceutically acceptable salts and solvates thereof, wherein R1, R2, R3, R4, R5, R6, R7, R8, R9, and R10 have the meanings as indicated in the specification, are useful for treating diseases mediated by blockade of the epithelial sodium channel. Pharmaceutical compositions that contain the compounds and processes for preparing the compounds are also described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.