Process for the preparation of aliskiren

US9056816B2 · kind B2 · utility

Assignee

• Jubilant Life Sciences Limited · IN

Inventors

• Sujay Biswas · New Delhi, IN
• Sankareswaran Srimurugan · Sidhauli, IN
• Anjul Kumar · Sidhauli, IN
• Atulya Kumar Panda · Sidhauli, IN
• Danish Jamshad · Nakodar, IN
• Mukesh Masand · Sidhauli, IN
• Bidyut Biswas · Sidhauli, IN
• Vikas Bansal · Sidhauli, IN
• Ashish Gupta · Houston, US
• Dharam Vir · Sidhauli, IN

Key dates

• Filing date: Oct 19, 2012
• Grant date: Jun 16, 2015
• Expiry date: Oct 19, 2032

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D307/33
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

The present invention provides a novel process and novel intermediates useful in the synthesis of pharmaceutically active compounds, especially renin inhibitors, such as Aliskiren, or a salt thereof, preferably Aliskiren hemifumarate.