Tetrahydrophenanthridinones and tetrahydrocyclopentaquinolinones as parp and tubulin polymerization inhibitors
US9150540B2 · kind B2 · utility
1Cited by
14References
8Claims
0Family size
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Key dates
| Filing date | Oct 14, 2014 |
| Grant date | Oct 6, 2015 |
| Priority date | — |
| Expiry date | Oct 14, 2034 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D221/12
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The present invention provides compounds of formula (I), their use as inhibitors of tubulin polymerization and their use as PARP inhibitors as well as pharmaceutical compositions comprising said compounds of formula (I)wherein R1, R2, R3, R4, R5, R6, R7 and Y have defined meanings.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.