Patent · US Active

Ester derivatives of androgen receptor modulators and methods for their use

US9173939B2 · kind B2 · utility

16Cited by
15References
29Claims
0Family size

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Key dates

Filing dateMay 9, 2014
Grant dateNov 3, 2015
Priority date
Expiry dateMay 9, 2034

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds having a structure of Structure I:or a pharmaceutically acceptable salt, tautomer, or stereoisomer thereof, wherein R1, R2, R3, R4, R5, J1, J2, X, Z, n1 and n2 are as defined herein, and wherein at least one of R1, R2 or R3 is an alkyl, alkenyl, aryl or aralkyl ester, are provided. Uses of such compounds for treatment of various indications, including prostate cancer, as well as methods of treatment involving such compounds are also provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.