Tubulysins and processes for preparing
US9187521B2 · kind B2 · utility
2Cited by
71References
29Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Oct 23, 2008 |
| Grant date | Nov 17, 2015 |
| Priority date | — |
| Expiry date | Jan 8, 2030 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07K5/06139
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Processes are described for the preparation of tubulysins. The processes are useful for preparing predetermined mixtures of tubulysins, preparing single tubulysins from mixtures of tubulysins, and for converting one tubulysin into a different tubulysin. The tubulysins described herein are useful in treating diseases and disease states that include pathogenic cell populations.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.