Patent · US Active

Folate receptor binding conjugates of antifolates

US9192682B2 · kind B2 · utility

13Cited by
3References
15Claims
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Key dates

Filing dateAug 26, 2013
Grant dateNov 24, 2015
Priority date
Expiry dateAug 26, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Conjugates of antifolates, releasable linkers, and drugs, and pharmaceutical compositions containing them are described. The conjugates are useful for treating diseases arising from pathogenic cell populations. Methods for treating such diseases are also described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.