Patent · US Active

Thieno[3,2-c]pyridine potassium channel inhibitors

US9216992B2 · kind B2 · utility

0Cited by
12References
11Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 8, 2006
Grant dateDec 22, 2015
Priority date
Expiry dateJan 6, 2030

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention provides thienopyridine compounds which are potassium channel inhibitors. In another embodiment, the invention provides pharmaceutical compositions comprising thienopyridines. In another embodiment, the invention provides methods of using thienopyridines in the treatment or prevention of cancer, arrhythmias, autoimmune diseases and inflammatory diseases, including gastric cancer, atrial fibrillation, type-2 diabetes mellitus, rheumatoid arthritis, type-1 diabetes, inflammatory bowel disorder and demyelinating disorders such as multiple sclerosis.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.