Patent · US Active

1,4-dihydro-naphthyridine derivative and pharmaceutical composition and use thereof

US9284330B2 · kind B2 · utility

0Cited by
0References
6Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 7, 2012
Grant dateMar 15, 2016
Priority date
Expiry dateDec 7, 2032

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D491/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed are 1,4-dihydro-naphthyridine derivatives and pharmaceutical composition and uses thereof. The 1,4-dihydro-naphthyridine derivatives are a compound capable of inhibiting acetylcholinesterase activity and preventing extracellular calcium from flowing into a cell via a calcium channel, i.e., having a dual-activity, which are of potential importance as a pharmaceutical and can be used to prepare the drugs for treating cardiovascular diseases, cerebrovascular diseases and dementia.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.