Patent · US Active

Pyrazolopyrimidines and related heterocycles as CK2 inhibitors

US9303033B2 · kind B2 · utility

6Cited by
1References
44Claims
0Family size

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Key dates

Filing dateSep 13, 2013
Grant dateApr 5, 2016
Priority date
Expiry dateSep 13, 2033

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides compounds that inhibit protein kinase CK2 activity (CK2 activity), and compositions containing such compounds. These compounds and compositions are useful for treating proliferative disorders such as cancer, as well as other kinase-associated conditions including inflammation, pain, and certain immunological disorders, and have the following general formula:

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.