Patent · US Active

Solid forms of nilotinib hydrochloride

US9376419B2 · kind B2 · utility

6Cited by
0References
18Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 15, 2013
Grant dateJun 28, 2016
Priority date
Expiry dateOct 15, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/13
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Disclosed are solid forms of Nilotinib hydrochloride and methods of preparation of various crystalline solvates of Nilotinib HCl including benzyl alcohol, acetic acid, propylene glycol, and isopropanol. Nilotinib HCl is a tyrosine kinase inhibitor used for the treatment of drug resistant chronic myelogenous leukemia (CML).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.