Bisphenol derivatives and their use as androgen receptor activity modulators
US9388112B2 · kind B2 · utility
14Cited by
17References
34Claims
0Family size
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Key dates
| Filing date | Jan 6, 2011 |
| Grant date | Jul 12, 2016 |
| Priority date | — |
| Expiry date | May 26, 2032 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D401/06
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
This invention provides bisphenol derivatives having a structure of formula 1. Said compounds are modulators of the androgen receptor activity and are useful in the treatment of various diseases, including prostate cancer, breast cancer, ovarian cancer, endometrial cancer, acne, ovarian cysts, polycystic ovarian disease, age-related macular degeneration, precocious puberty, hirsutism and hair loss.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.