Patent · US Active

Process for producing optically active succinimide derivatives and intermediates thereof

US9434737B2 · kind B2 · utility

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Key dates

Filing dateDec 12, 2013
Grant dateSep 6, 2016
Priority date
Expiry dateJan 23, 2034

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07B2200/07
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

Provided is a process for producing (3R)-2′-(4-bromo-2-fluorobenzyl)spiro{pyrrolidine-3,4′(1′H)-pyrrolo[1,2-a]pyrazine}-1′,2,3′,5(2′H)-tetraone (compound A). The method includes converting an optically active succinimide derivative of formula (I) to compound A, in which the compound of formula (I) has been prepared by reacting a base with an optically active amide derivative of formula (VI).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.