Patent · US Active

Spirocyclic dihydro-thiazine and dihydro-oxazine BACE inhibitors, and compositions and uses thereof

US9493485B2 · kind B2 · utility

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19Claims
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Assignee

Inventors

Key dates

Filing dateMar 20, 2013
Grant dateNov 15, 2016
Priority date
Expiry dateMar 20, 2033

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D498/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds are provided having a structure according to Formula (I): wherein A1, A2, A3, Y, R1, R2, R3, R4, R5, R6, m, n and p are defined herein. Further provided are pharmaceutical compositions including the compounds provided and methods of making and using the compounds and compositions as provided, e.g., in the treatment and prevention of various disorders, such as Alzheimer's disease.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.