Patent · US Active

N-containing heterocyclic compounds

US9499560B2 · kind B2 · utility

2Cited by
3References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 15, 2014
Grant dateNov 22, 2016
Priority date
Expiry dateMay 16, 2034

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to N-containing heterocyclic compounds that are inhibitors of protein kinases including JAK kinases. In particular, the compounds are selective for JAK1, JAK2, JAK3 or TYK2 kinases and combinations thereof such as JAK1 and JAK2. The kinase inhibitors can be used in the treatment of kinase associated diseases such as immunological and inflammatory diseases including organ transplants; hyperproliferative diseases including cancer and myeloproliferative diseases; viral diseases; metabolic diseases; and vascular diseases.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.