Patent · US Active

Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes

US9517228B2 · kind B2 · utility

7Cited by
9References
18Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 3, 2015
Grant dateDec 13, 2016
Priority date
Expiry dateSep 3, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D231/06
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides novel, diastereomeric pyrazolines that are useful as cannabinoid receptor blockers and pharmaceutical compositions thereof and methods of using the same for treating obesity, diabetes, inflammatory disorders, cardiometabolic disorders, hepatic disorders, and/or cancers.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.