Patent · US Active

Folate receptor binding conjugates of antifolates

US9549992B2 · kind B2 · utility

5Cited by
3References
1Claims
0Family size

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Key dates

Filing dateOct 21, 2015
Grant dateJan 24, 2017
Priority date
Expiry dateOct 21, 2035

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Conjugates of antifolates, releasable linkers, and drugs, and pharmaceutical compositions containing them are described. The conjugates are useful for treating diseases arising from pathogenic cell populations. Methods for treating such diseases are also described.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.