Patent · US Active

Binding ligand linked drug delivery conjugates of tubulysins

US9555139B2 · kind B2 · utility

0Cited by
127References
15Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 13, 2008
Grant dateJan 31, 2017
Priority date
Expiry dateJun 15, 2029

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07K5/06078
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Described herein are compounds, pharmaceutical compositions and methods for treating pathogenic cell populations. The compounds described herein include conjugates of tubulysins and vitamin receptor binding ligands. The conjugates also include a releasable bivalent linker.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.