2-acylaminothiazole derivative or salt thereof
US9562044B2 · kind B2 · utility
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16Claims
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Key dates
| Filing date | Feb 27, 2014 |
| Grant date | Feb 7, 2017 |
| Priority date | — |
| Expiry date | Feb 27, 2034 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D491/107
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Thiazole derivatives having pyrazine-2-carbonylamino substituted at the 2-position of the following formula (I):are excellent muscarinic M3 receptor positive allosteric modulators, and are useful for treating bladder or urinary tract diseases, related to bladder contraction by a muscarinic M3 receptor. The 2-acylaminothiazole derivatives and salts thereof can be used for treating bladder or urinary tract diseases, related to bladder contraction by a muscarinic M3 receptor, for example, voiding dysfunctions such as underactive bladder.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.