Patent · US Active

Cell-targeting nanoparticles comprising polynucleotide agents and uses thereof

US9574210B2 · kind B2 · utility

3Cited by
24References
36Claims
0Family size

Assignee

Inventor

Key dates

Filing dateJul 29, 2010
Grant dateFeb 21, 2017
Priority date
Expiry dateJul 29, 2030

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY10T428/2991
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A method of generating a particle is disclosed, the particle being for delivery of a polynucleotide to a target cell. The method comprises (a) contacting the polynucleotide with a composition comprising cationic molecules, wherein the cationic molecules condense the polynucleotide by electrostatic interactions to generate a complex, wherein the cationic molecules are not comprised in a liposome; and (b) covalently binding the complex to a targeting moiety at a pH equal to or below about 4.5, thereby generating the particle for delivery of the polynucleotide agent to the target cell. Use of the particles and compositions comprising same are also disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.